MAP3K15

Mitogen-activated protein kinase kinase kinase 1 UniProt accession Q13233

Component of a protein kinase signal transduction cascade (PubMed:9808624). Activates the ERK and JNK kinase pathways by phosphorylation of MAP2K1 and MAP2K4 (PubMed:9808624). May phosphorylate the MAPK8/JNK1 kinase (PubMed:17761173).

Activates CHUK and IKBKB, the central protein kinases of the NF-kappa-B pathway (PubMed:9808624)

Source: UniProt

Binds both upstream activators and downstream substrates in multimolecular complexes through its N-terminus (PubMed:9808624). Oligomerizes after binding MAP2K4 or TRAF2 (PubMed:9808624). Interacts with AXIN1 (PubMed:12223491, PubMed:15262978).

Interacts (via the kinase catalytic domain) with STK38 (PubMed:17906693). Interacts with GRIPAP1 (PubMed:17761173)

Source: UniProt
  • 46,XY sex reversal 6 (SRXY6)

    A disorder of sex development. Affected individuals have a 46,XY karyotype but present as phenotypically normal females.

Source: UniProt

Click a pathway to open the interactive Reactome viewer.

Pathway list and interactive viewer: Reactome

Synthetic Lethal Network

Genes with an experimentally identified or computationally predicted synthetic-lethal relationship to MAP3K15, aggregated across our SSL data sources. Click any partner node to view that gene’s page.

Nodes and edges are coloured by the SSL data source. Partners appearing in more than one source are shown in grey.

BioGRID SLOrth SynLethDB MexDrugs Multi-source
Sources: BioGRID, SLOrth, SynLethDB, MexDrugs

Clinical Trials

Total Trials Found: 32

NCT ID Condition Brief Title Phase Status
NCT03176485 Metastatic Cancer, Melanoma, Colon Cancer, Differentiated Thyroid Cancer, Hepatocellular Carcinoma, Renal Cell Carcinoma, Metastatic Melanoma, HCC, Metastatic Colon Cancer Evaluation of Pathway Modulation by Raf, MEK, & Kinase Inhibitors NA COMPLETED
NCT03416933 Melanoma (Skin) Therapeutic Drug Monitoring of BRAF-mutated Advanced Melanoma NA COMPLETED
NCT06555237 Cardiomegaly, Noonan Syndrome MEK Inhibitors for the Treatment of Hypertrophic Cardiomyopathy in Patients With RASopathies PHASE2 RECRUITING